BDBM60917 9-chloranyl-5-(4-hydroxyphenyl)-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol;methanesulfonic acid::9-chloro-5-(4-hydroxyphenyl)-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol;mesylic acid::9-chloro-5-(4-hydroxyphenyl)-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol;methanesulfonic acid::FENOLDOPAM::FENOLDOPAM MESYLATE::MLS001401388::SMR000469190::cid_49659
SMILES Oc1ccc(cc1)C1CNCCc2c(Cl)c(O)c(O)cc12
InChI Key InChIKey=TVURRHSHRRELCG-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 60917
Affinity DataKi: 13nMAssay Description:Binding affinity against Dopamine receptor D2 in rat striatal membranes using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Compound was tested for inhibition of [3H]spiroperidol binding against Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+4nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Displacement of [3H]-spiroperidol from homogenized bovine pituitary Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair